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Items: 1 to 20 of 229

1.

Structure-function of the G protein-coupled receptor superfamily.

Katritch V, Cherezov V, Stevens RC.

Annu Rev Pharmacol Toxicol. 2013;53:531-56. doi: 10.1146/annurev-pharmtox-032112-135923. Epub 2012 Nov 8. Review.

2.

Conformational analysis of g protein-coupled receptor signaling by hydrogen/deuterium exchange mass spectrometry.

Li S, Lee SY, Chung KY.

Methods Enzymol. 2015;557:261-78. doi: 10.1016/bs.mie.2014.12.004. Epub 2015 Mar 29.

PMID:
25950969
3.

Agonist-induced conformational changes in bovine rhodopsin: insight into activation of G-protein-coupled receptors.

Bhattacharya S, Hall SE, Vaidehi N.

J Mol Biol. 2008 Oct 3;382(2):539-55. doi: 10.1016/j.jmb.2008.06.084. Epub 2008 Jul 7.

PMID:
18638482
4.

Structural basis for ligand binding and specificity in adrenergic receptors: implications for GPCR-targeted drug discovery.

Huber T, Menon S, Sakmar TP.

Biochemistry. 2008 Oct 21;47(42):11013-23. doi: 10.1021/bi800891r. Epub 2008 Sep 27.

PMID:
18821775
5.

The Molecular Basis of G Protein-Coupled Receptor Activation.

Weis WI, Kobilka BK.

Annu Rev Biochem. 2018 Jun 20;87:897-919. doi: 10.1146/annurev-biochem-060614-033910. Review.

6.

Allosteric modulation of G-protein coupled receptors.

Jensen AA, Spalding TA.

Eur J Pharm Sci. 2004 Mar;21(4):407-20. Review.

PMID:
14998571
7.

G-protein-coupled receptor structure, ligand binding and activation as studied by solid-state NMR spectroscopy.

Ding X, Zhao X, Watts A.

Biochem J. 2013 Mar 15;450(3):443-57. doi: 10.1042/BJ20121644. Review. Erratum in: Biochem J. 2013 Apr 15;451(2):343.

PMID:
23445222
9.

GPCR crystal structures: Medicinal chemistry in the pocket.

Shonberg J, Kling RC, Gmeiner P, Löber S.

Bioorg Med Chem. 2015 Jul 15;23(14):3880-906. doi: 10.1016/j.bmc.2014.12.034. Epub 2014 Dec 24. Review.

PMID:
25638496
10.

Emerging structural insights into biased GPCR signaling.

Shukla AK, Singh G, Ghosh E.

Trends Biochem Sci. 2014 Dec;39(12):594-602. doi: 10.1016/j.tibs.2014.10.001. Epub 2014 Nov 4. Review.

PMID:
25458114
11.

Conformational changes of G protein-coupled receptors during their activation by agonist binding.

Bissantz C.

J Recept Signal Transduct Res. 2003;23(2-3):123-53. Review.

PMID:
14626443
12.

Signaling within Allosteric Machines: Signal Transmission Pathways Inside G Protein-Coupled Receptors.

Bartuzi D, Kaczor AA, Matosiuk D.

Molecules. 2017 Jul 15;22(7). pii: E1188. doi: 10.3390/molecules22071188. Review.

13.

Structural insights into ligand recognition and selectivity for classes A, B, and C GPCRs.

Lee SM, Booe JM, Pioszak AA.

Eur J Pharmacol. 2015 Sep 15;763(Pt B):196-205. doi: 10.1016/j.ejphar.2015.05.013. Epub 2015 May 14. Review.

14.

Ligand-stabilized conformational states of human beta(2) adrenergic receptor: insight into G-protein-coupled receptor activation.

Bhattacharya S, Hall SE, Li H, Vaidehi N.

Biophys J. 2008 Mar 15;94(6):2027-42. Epub 2007 Dec 7.

15.

A conformation-equilibrium model captures ligand-ligand interactions and ligand-biased signalling by G-protein coupled receptors.

Roth S, Bruggeman FJ.

FEBS J. 2014 Oct;281(20):4659-71. doi: 10.1111/febs.12970. Epub 2014 Sep 17.

16.

SnapShot: GPCR-Ligand Interactions.

Ghosh E, Nidhi K, Shukla AK.

Cell. 2014 Dec 18;159(7):1712, 1712.e1. doi: 10.1016/j.cell.2014.12.008.

17.

Emerging opportunities for allosteric modulation of G-protein coupled receptors.

Wang CI, Lewis RJ.

Biochem Pharmacol. 2013 Jan 15;85(2):153-62. doi: 10.1016/j.bcp.2012.09.001. Epub 2012 Sep 11. Review.

PMID:
22975406
18.

Structural and biophysical characterisation of G protein-coupled receptor ligand binding using resonance energy transfer and fluorescent labelling techniques.

Ward RJ, Milligan G.

Biochim Biophys Acta. 2014 Jan;1838(1 Pt A):3-14. doi: 10.1016/j.bbamem.2013.04.007. Epub 2013 Apr 13. Review.

19.

Diversity and modularity of G protein-coupled receptor structures.

Katritch V, Cherezov V, Stevens RC.

Trends Pharmacol Sci. 2012 Jan;33(1):17-27. doi: 10.1016/j.tips.2011.09.003. Epub 2011 Oct 25. Review.

20.

Structural insights into agonist-induced activation of G-protein-coupled receptors.

Deupi X, Standfuss J.

Curr Opin Struct Biol. 2011 Aug;21(4):541-51. doi: 10.1016/j.sbi.2011.06.002. Epub 2011 Jun 30. Review.

PMID:
21723721

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