Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Binding affinity towards human ADRA1A in an in vitro assay with cellular components (NIBR assay) measured by scintillation proximity assay
Assay data:49 Active, 29 Activity ≤ 1 µM, 231 Tested
SummaryRelated BioAssays by Target
Antagonist activity at human ADRA1A in an in vitro cell-based assay measured by fluorescence spectroscopy
Assay data:117 Active, 53 Activity ≤ 1 µM, 881 Tested
Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting
Assay data:176 Active, 1 Activity ≤ 1 nM, 87 Activity ≤ 1 µM, 1215 Tested
Binding affinity towards human HTR1A in an in vitro assay with cellular components measured by scintillation counting
Assay data:56 Active, 33 Activity ≤ 1 µM, 377 Tested
Binding affinity towards human ADRA2A in an in vitro assay with cellular components measured by scintillation counting
Assay data:63 Active, 20 Activity ≤ 1 µM, 323 Tested
Binding affinity towards human TACR1 in an in vitro assay with cellular components measured by membrane filtration
Assay data:19 Active, 4 Activity ≤ 1 µM, 218 Tested
Binding affinity towards human HTR2B in an in vitro assay with cellular components measured by membrane filtration
Assay data:103 Active, 70 Activity ≤ 1 µM, 317 Tested
Antagonist activity at human HTR2B in an in vitro cell-based assay measured by fluorescent imaging plate reader
Assay data:147 Active, 45 Activity ≤ 1 µM, 1167 Tested
Binding affinity towards human HTR2A in an in vitro assay with cellular components measured by membrane filtration
Assay data:140 Active, 4 Activity ≤ 1 nM, 75 Activity ≤ 1 µM, 414 Tested
Agonist activity at human HTR1A in an in vitro cell-based assay measured by fluorescent imaging plate reader
Assay data:41 Active, 16 Activity ≤ 1 µM, 1178 Tested
Binding affinity towards human DRD4 in an in vitro assay with cellular components measured by membrane filtration
Assay data:36 Active, 19 Activity ≤ 1 µM, 233 Tested
Binding affinity towards human DRD2 in an in vitro assay with cellular components measured by membrane filtration, scintillation proximity assay
Assay data:153 Active, 2 Activity ≤ 1 nM, 73 Activity ≤ 1 µM, 1228 Tested
Binding affinity towards human AGTR1 in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:26 Active, 5 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 1184 Tested
Binding affinity towards human ADRB3 in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:17 Active, 3 Activity ≤ 1 µM, 299 Tested
Binding affinity towards human ADRB2 in an in vitro assay with cellular components measured by radioactivity method
Assay data:58 Active, 21 Activity ≤ 1 µM, 952 Tested
Compound was evaluated for inhibition of human ADRB1 in an in vitro assay measured by radioactivity method
Assay data:66 Active, 1 Activity ≤ 1 nM, 26 Activity ≤ 1 µM, 1195 Tested
Compound was evaluated for inhibition of human ADRA2C in an in vitro assay with cellular components measured by membrane filtration
Assay data:195 Active, 66 Activity ≤ 1 µM, 1241 Tested
Binding affinity towards human ADRA2B in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:166 Active, 1 Activity ≤ 1 nM, 62 Activity ≤ 1 µM, 1209 Tested
Assay data:150 Active, 65 Activity ≤ 1 µM, 699 Tested
3H-CGP 12177 Whole Cell Binding Assay from Article 10.1038/sj.bjp.0706048: "The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors."
Assay data:25 Active, 7 Activity ≤ 1 nM, 23 Activity ≤ 1 µM, 25 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on