BioAssays, Active for PubChem Compound (Select 2585) - PubChem BioAssay - NCBI

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Select item 19618681.

Binding affinity towards human ADRA1A in an in vitro assay with cellular components (NIBR assay) measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Alpha-1A adrenergic receptor

Assay data:49 Active, 29 Activity ≤ 1 µM, 231 Tested

AID:: 1961868

Summary Related BioAssays by Target

Select item 19618592.

Binding affinity towards human DRD1 in an in vitro assay with cellular components (NIBR assay) measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(1A) dopamine receptor

Assay data:35 Active, 19 Activity ≤ 1 µM, 305 Tested

AID:: 1961859

Summary Related BioAssays by Target

Select item 19618583.

Antagonist activity at human ADRA1A in an in vitro cell-based assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Alpha-1A adrenergic receptor

Assay data:117 Active, 53 Activity ≤ 1 µM, 881 Tested

AID:: 1961858

Summary Related BioAssays by Target

Select item 19618564.

Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(3) dopamine receptor

Assay data:176 Active, 1 Activity ≤ 1 nM, 87 Activity ≤ 1 µM, 1215 Tested

AID:: 1961856

Summary Related BioAssays by Target

Select item 19618535.

Binding affinity towards human HTR1A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1A

Assay data:56 Active, 33 Activity ≤ 1 µM, 377 Tested

AID:: 1961853

Summary Related BioAssays by Target

Select item 19618516.

Binding affinity towards human OPRM1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Mu-type opioid receptor

Assay data:60 Active, 9 Activity ≤ 1 µM, 766 Tested

AID:: 1961851

Summary Related BioAssays by Target

Select item 19618507.

Binding affinity towards human ADRA2A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Alpha-2A adrenergic receptor

Assay data:63 Active, 20 Activity ≤ 1 µM, 323 Tested

AID:: 1961850

Summary Related BioAssays by Target

Select item 19618498.

Binding affinity towards human SLC6A4 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:148 Active, 75 Activity ≤ 1 µM, 1194 Tested

AID:: 1961849

Summary Related BioAssays by Target

Select item 19618489.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:123 Active, 40 Activity ≤ 1 µM, 1197 Tested

AID:: 1961848

Summary Related BioAssays by Target

Select item 196184710.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:119 Active, 21 Activity ≤ 1 µM, 1213 Tested

AID:: 1961847

Summary Related BioAssays by Target

Select item 196184111.

Binding affinity towards human TACR1 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: Substance-P receptor

Assay data:19 Active, 4 Activity ≤ 1 µM, 218 Tested

AID:: 1961841

Summary Related BioAssays by Target

Select item 196183512.

Compound was evaluated for inhibition of human SCN5A in an in vitro cell-based assay measured by IonWorks automated patch clamp

Source:: ChEMBL

Protein Target:: Sodium channel protein type 5 subunit alpha

Assay data:37 Active, 5 Activity ≤ 1 µM, 230 Tested

AID:: 1961835

Summary Related BioAssays by Target

Select item 196181113.

Agonist activity at human OPRM1 in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Mu-type opioid receptor

Assay data:43 Active, 9 Activity ≤ 1 µM, 711 Tested

AID:: 1961811

Summary Related BioAssays by Target

Select item 196180314.

Binding affinity towards human NR1I2 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: Nuclear receptor subfamily 1 group I member 2

Assay data:101 Active, 19 Activity ≤ 1 µM, 846 Tested

AID:: 1961803

Summary Related BioAssays by Target

Select item 196180115.

Agonist activity at human NR1I2 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: Nuclear receptor subfamily 1 group I member 2

Assay data:41 Active, 11 Activity ≤ 1 µM, 580 Tested

AID:: 1961801

Summary Related BioAssays by Target

Select item 196179016.

Binding affinity towards human MLNR in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Motilin receptor

Assay data:28 Active, 3 Activity ≤ 1 µM, 1179 Tested

AID:: 1961790

Summary Related BioAssays by Target

Select item 196178517.

Compound was evaluated for inhibition of human KCNH2 in an in vitro assay with cellular components measured by membrane filtration, radioactivity method

Source:: ChEMBL

Protein Target:: Potassium voltage-gated channel subfamily H member 2

Assay data:353 Active, 116 Activity ≤ 1 µM, 1804 Tested

AID:: 1961785

Summary Related BioAssays by Target

Select item 196178418.

Binding affinity towards human HTR7 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 7

Assay data:19 Active, 10 Activity ≤ 1 µM, 144 Tested

AID:: 1961784

Summary Related BioAssays by Target

Select item 196178319.

Binding affinity towards human HTR6 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 6

Assay data:27 Active, 15 Activity ≤ 1 µM, 148 Tested

AID:: 1961783

Summary Related BioAssays by Target

Select item 196178020.

Binding affinity towards human HTR2C in an in vitro assay with cellular components measured by radioactivity method

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2C

Assay data:123 Active, 1 Activity ≤ 1 nM, 48 Activity ≤ 1 µM, 1199 Tested

AID:: 1961780

Summary Related BioAssays by Target

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Proteins (23)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (99)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (27)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (58)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (15)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

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BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (78)
BioAssays extracted from the literature
NIH MLP (23)
BioAssays deposited by the NIH Molecular Libraries Program
Other (33)
BioAssays deposited by other experimentalists

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