BioAssays, Active for PubChem Compound (Select 162642759) - PubChem BioAssay - NCBI

Warning: The NCBI web site requires JavaScript to function. more...

Links from PubChem Compound

Items: 1 to 20 of 34

<< First< Prev

Page of 2

Select item 18951411.

Inhibition of GST-tagged human SIK2 autophosphorylation measured after 30 mins in presence of [gamma33P]ATP by Western blot analysis

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase SIK2

Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1895141

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18951382.

Inhibition of full length C-terminal nanoLuc-tagged human TIE2 expressed in HEK293 cells using NanoBRET NanoGlo substrate incubated for 2 hrs in presence of tracer K10 by NanoBRET assay

Source:: ChEMBL

Protein Target:: Angiopoietin-1 receptor

Assay data:1 Active, 1 Tested

AID:: 1895138

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951353.

Inhibition of full length C-terminal nanoLuc-tagged human PKN3 expressed in HEK293 cells using NanoBRET NanoGlo substrate incubated for 2 hrs in presence of tracer K10 by NanoBRET assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N3

Assay data:1 Active, 1 Tested

AID:: 1895135

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951344.

Inhibition of full length C-terminal nanoLuc-tagged human NLK expressed in HEK293 cells using NanoBRET NanoGlo substrate incubated for 2 hrs in presence of tracer K10 by NanoBRET assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase NLK

Assay data:1 Active, 1 Tested

AID:: 1895134

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951305.

Inhibition of full length N-terminal nanoLuc-tagged human SIK1 expressed in HEK293 cells using NanoBRET NanoGlo substrate incubated for 2 hrs in presence of tracer K10 by NanoBRET assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase SIK1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895130

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18951296.

Inhibition of human MELK by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Maternal embryonic leucine zipper kinase

Assay data:1 Active, 1 Tested

AID:: 1895129

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951287.

Inhibition of human MST4 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 26

Assay data:1 Active, 1 Tested

AID:: 1895128

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951278.

Inhibition of human TIE2 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Angiopoietin-1 receptor

Assay data:1 Active, 1 Tested

AID:: 1895127

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18951269.

Inhibition of human MAP2K4 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Dual specificity mitogen-activated protein kinase kinase 4

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895126

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189512510.

Inhibition of human PAK1 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase PAK 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895125

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189512411.

Inhibition of human PKN3 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N3

Assay data:1 Active, 1 Tested

AID:: 1895124

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 189512312.

Inhibition of human NLK by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase NLK

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895123

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189512213.

Inhibition of human PAK2 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase PAK 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895122

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189512114.

Inhibition of human PAK3 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase PAK 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895121

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189512015.

Inhibition of human MAP4K5 (KHS1) by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895120

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189511916.

Inhibition of human SIK1 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase SIK1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895119

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189511817.

Inhibition of human SIK3 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase SIK3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895118

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189511718.

Inhibition of human SIK2 by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase SIK2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895117

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189515319.

Antitumor activity in human HeLa cells cultured as 3D spheroids assessed as increase in dead cells at 5 uM incubated for 48 hrs in presence of paclitaxel by immunofluorescence analysis

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895153

Summary Compounds, Active PubMed Citation

Select item 189515220.

Antitumor activity in human HeLa cells cultured as 3D spheroids assessed as increase in dead cells at 5 uM incubated for 48 hrs by immunofluorescence analysis

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895152

Summary Compounds, Active PubMed Citation

<< First< Prev

Page of 2

Supplemental Content

Filters: Manage Filters

Refine your results

• What's this?

BioActivity

Active Compounds (34)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (1)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (16)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (23)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (5)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Depositor Category

Literature Extraction (24)
BioAssays extracted from the literature
Other (10)
BioAssays deposited by other experimentalists

Actions on your results

View or Download BioAssay in PubChem

Find related data

Recent activity

Clear Turn Off Turn On

BioAssays, Active for PubChem Compound (Select 162642759) (34)
PubChem BioAssay

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...

You are here: NCBI > Chemicals & Bioassays > PubChem BioAssay