BioAssays for PubChem Compound (Select 285033) - PubChem BioAssay - NCBI

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Select item 19620161.

Cytotoxicity activity against human HepG2 cells assessed by CellTiter-Glo luminescent cell viability assay.

Source:: ChEMBL

Assay data:1241 Active, 184 Activity ≤ 1 µM, 1545 Tested

AID:: 1962016

Select item 19618452.

Antagonist activity at human TBXA2R in an in vitro cell-based assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:34 Active, 15 Activity ≤ 1 µM, 906 Tested

AID:: 1961845

Summary Related BioAssays by Target

Select item 19618443.

Agonist activity at human TBXA2R in an in vitro cell-based assay (CRO assay) measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:13 Active, 8 Activity ≤ 1 µM, 927 Tested

AID:: 1961844

Summary Related BioAssays by Target

Select item 19618404.

Binding affinity towards human SLC6A4 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:99 Active, 36 Activity ≤ 1 µM, 927 Tested

AID:: 1961840

Summary Related BioAssays by Target

Select item 19618395.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:128 Active, 38 Activity ≤ 1 µM, 927 Tested

AID:: 1961839

Summary Related BioAssays by Target

Select item 19618386.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:137 Active, 27 Activity ≤ 1 µM, 927 Tested

AID:: 1961838

Summary Related BioAssays by Target

Select item 19618287.

Compound was evaluated for inhibition of human PTGS1 in an in vitro cell free assay measured by fluorescence method

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 1

Assay data:80 Active, 33 Activity ≤ 1 µM, 924 Tested

AID:: 1961828

Summary Related BioAssays by Target

Select item 19618268.

Compound was evaluated for inhibition of human PTGS1 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 1

Assay data:96 Active, 35 Activity ≤ 1 µM, 927 Tested

AID:: 1961826

Summary Related BioAssays by Target

Select item 19618209.

Binding affinity towards human PGR in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Progesterone receptor

Assay data:87 Active, 51 Activity ≤ 1 µM, 927 Tested

AID:: 1961820

Summary Related BioAssays by Target

Select item 196181410.

Compound was evaluated for inhibition of human PDE4A in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A

Assay data:46 Active, 10 Activity ≤ 1 µM, 927 Tested

AID:: 1961814

Summary Related BioAssays by Target

Select item 196181311.

Compound was evaluated for inhibition of human PDE3A in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: cGMP-inhibited 3',5'-cyclic phosphodiesterase A

Assay data:15 Active, 6 Activity ≤ 1 µM, 927 Tested

AID:: 1961813

Summary Related BioAssays by Target

Select item 196181212.

Binding affinity towards human OPRM1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Mu-type opioid receptor

Assay data:117 Active, 24 Activity ≤ 1 µM, 927 Tested

AID:: 1961812

Summary Related BioAssays by Target

Select item 196178713.

Compound was evaluated for inhibition of human MAOA in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Amine oxidase [flavin-containing] A

Assay data:13 Active, 5 Activity ≤ 1 µM, 927 Tested

AID:: 1961787

Summary Related BioAssays by Target

Select item 196178514.

Compound was evaluated for inhibition of human KCNH2 in an in vitro assay with cellular components measured by membrane filtration, radioactivity method

Source:: ChEMBL

Protein Target:: Potassium voltage-gated channel subfamily H member 2

Assay data:353 Active, 116 Activity ≤ 1 µM, 1804 Tested

AID:: 1961785

Summary Related BioAssays by Target

Select item 196177715.

Agonist activity at human HTR2B in an in vitro cell-based assay (CRO assay) measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2B

Assay data:3 Active, 5 Activity ≤ 1 µM, 927 Tested

AID:: 1961777

Summary Related BioAssays by Target

Select item 196177216.

Binding affinity towards human HTR1A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1A

Assay data:141 Active, 68 Activity ≤ 1 µM, 927 Tested

AID:: 1961772

Summary Related BioAssays by Target

Select item 196176917.

Binding affinity towards human HRH3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Histamine H3 receptor

Assay data:23 Active, 11 Activity ≤ 1 µM, 927 Tested

AID:: 1961769

Summary Related BioAssays by Target

Select item 196175718.

Binding affinity towards rat Gabra1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Gamma-aminobutyric acid receptor subunit alpha-1

Assay data:6 Active, 1 Activity ≤ 1 µM, 532 Tested

AID:: 1961757

Summary Related BioAssays by Target

Select item 196175119.

Compound was evaluated for inhibition of human F2 in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Prothrombin

Assay data:11 Active, 8 Activity ≤ 1 µM, 927 Tested

AID:: 1961751

Summary Related BioAssays by Target

Select item 196174920.

Binding affinity towards human ESR1 in an in vitro cell free assay (CRO assay) measured by membrane filtration

Source:: ChEMBL

Protein Target:: Estrogen receptor

Assay data:31 Active, 1 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 927 Tested

AID:: 1961749

Summary Related BioAssays by Target

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Target

Proteins (202)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (454)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (57)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (174)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Confirmatory (344)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (125)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (191)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (117)
BioAssays extracted from the literature
NIH MLP (274)
BioAssays deposited by the NIH Molecular Libraries Program
Other (140)
BioAssays deposited by other experimentalists

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BioAssays for PubChem Compound (Select 285033) (564)
PubChem BioAssay
Profile neighbors for GEO Profiles (Select 47047558) (200)
GEO Profiles
ZMPSTE24 zinc metallopeptidase STE24 [Homo sapiens]
ZMPSTE24 zinc metallopeptidase STE24 [Homo sapiens]
Gene ID:10269

Gene
Gene Links for GEO Profiles (Select 28804687) (1)
Gene
Cdkn2aipnl CDKN2A interacting protein N-terminal like [Mus musculus]
Cdkn2aipnl CDKN2A interacting protein N-terminal like [Mus musculus]
Gene ID:52626

Gene

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