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CLK1 SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
CLK3 SGC Tm panel (DSF)
CLK1 Invitrogen Lab (UK) kinase screen (BI)
Inhibition of CLK2 (unknown origin) at 1 uM relative to control
Assay data:3 Tested
Inhibition of CLK1 (unknown origin) at 1 uM relative to control
Inhibition of CLK4 (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human CLK1 assessed as residence time measured upto 240 min by TR-FRET assay
Assay data:37 Tested
Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assay
Assay data:36 Active, 11 Activity ≤ 1 nM, 37 Activity ≤ 1 µM, 37 Tested
Inhibition of recombinant human CLK1 expressed in Sf9 insect cells using myelin basic protein as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay
Assay data:32 Active, 29 Activity ≤ 1 µM, 35 Tested
Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:45 Active, 40 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human CLK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:31 Active, 11 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human CLK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:46 Active, 1 Activity ≤ 1 nM, 27 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:45 Active, 37 Activity ≤ 1 µM, 56 Tested
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