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Antagonist activity at human NR1H4 in an in vitro cell free assay measured by luminescence method
Assay data:6 Active, 1 Activity ≤ 1 µM, 36 Tested
SummaryRelated BioAssays by Target
Antagonist activity at human NR1H4 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:3 Active, 36 Tested
Agonist activity at human NR1H4 in an in vitro cell free assay measured by luminescence method
Assay data:36 Tested
Agonist activity at human NR1H4 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:34 Tested
Agonist activity at FXR (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at full length FXR in human Huh-7 cells
Agonist activity at FXR (unknown origin) by fluorescence resonance energy tranfer assay
Activation of FXR (unknown origin) at 10 uM
Assay data:1 Active, 1 Tested
Partial agonist activity at FXR in human Huh-7 cells assessed as reduction in CDCA-induced SHP gene expression at 10 uM by RT-PCR analysis
Partial agonist activity at FXR in human Huh-7 cells assessed as reduction in CDCA-induced SREBP gene expression at 10 uM by RT-PCR analysis
Partial agonist activity at FXR in human Huh-7 cells assessed as reduction in CDCA-induced FAS gene expression at 10 uM by RT-PCR analysis
Partial agonist activity at FXR in human Huh-7 cells assessed as reduction in CDCA-induced OSTalpha gene expression at 10 uM by RT-PCR analysis
Partial agonist activity at FXR in human Huh-7 cells assessed as reduction in CDCA-induced BSEP gene expression at 10 uM by RT-PCR analysis
Antagonist activity at FXR-LBD-GST (unknown origin) in presence of GW4064 relative to control
Assay data:1 Tested
Antagonist activity at FXR-LBD-GST (unknown origin) in presence of GW4064
Assay data:1 Active, 2 Tested
Partial agonist activity at human FXR expressed in Huh-7 cells in presence of CDCA by luciferase reporter gene assay relative to GW4064
Assay data:2 Tested
Partial agonist activity at human FXR expressed in Huh-7 cells in presence of CDCA by luciferase reporter gene assay
Assay data:2 Active, 2 Tested
Partial agonist activity at FXR-LBD-GST (unknown origin) using fluorecein-SRC2-2 coactivator peptide by TR-FRET assay in relative to GW40
Assay data:9 Tested
Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assay
Assay data:9 Active, 9 Activity ≤ 1 µM, 18 Tested
Antagonist activity at FXR (unknown origin)
Assay data:3 Active, 3 Tested
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