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Inhibition of CK2 in mouse C2C12 cells assessed as reduction in CK2 substrates phosphorylation at 1 to 4 uM by Western blot analysis
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of CK2 in mouse C2C12 cells assessed as reduction in CDC37 phosphorylation at S13 residues at 1 to 4 uM by Western blot analysis
Inhibition of CK2 in mouse C2C12 cells assessed as reduction in Akt phosphorylation at S129 residues at 1 to 4 uM by Western blot analysis
Mouse Kv1.3 (Voltage-gated potassium channels)
Assay data:4 Active, 4 Tested
Inhibition of mouse Kv1.3 expressed in L929 cells at -80 mV holding potential by whole cell patch-clamp method
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [125I]-ChTX from mouse Kv1.3 after 20 mins by scintillation counting analysis
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Displacement of [3H]paroxetine from mouse SERT in whole brain membrane
Assay data:10 Active, 8 Activity ≤ 1 µM, 12 Tested
Inhibition of 5-HT transporter in NMRI albino mouse brain assessed as [3H]5-HT accumulation in hypothalamus after 5 mins
Assay data:5 Active, 2 Activity ≤ 1 µM, 6 Tested
Binding affinity to CSNK2A2 in mouse brain homogenate after 3 hrs by competition affinity chromatographic analysis
Binding affinity to CK2 alpha' subunit in mouse HT22 cell lysate by Western blot analysis
Assay data:1 Active, 1 Tested
Binding affinity to CK2 alpha' subunit in mouse brain homogenate by Western blot analysis
Displacement of [3H]-citalopram from SERT in mouse cortex after 2 hrs by liquid scintillation counting
Displacement of [3H]citalopram from mouse cortex SERT by filtration binding assay
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells at 10uM
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells
Assay data:55 Active, 23 Activity ≤ 1 µM, 57 Tested
Effective dose against potentiation of 5-HTP induced serotonin syndrome in mice upon oral administration (Serotonin reuptake inhibitory activity)
Assay data:22 Tested
Inhibition of Casein kinase 2 of P19 cells
Assay data:7 Tested
Effective concentration against murine voltage-gated potassium channel subunit Kv1.3 expressed in L929 cells using patch clamp
Assay data:1 Tested
Blockade of peak steady-state K+ currents of Kv1.3 channels in mice fibroblasts L929 at 50 uM
Assay data:2 Tested
Blockade of peak steady-state K+ currents of Kv1.3 channels in mice fibroblasts L929 at 25 uM
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