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Antagonist activity at recombinant human QRFP receptor expressed in CHO cells preincubated for 10 mins followed by agonist challenge in presence of probenecid by Fluo-4AM staining based fluorescence assay
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting method
Assay data:1 Active, 1 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
PRESTO-Tango GPCRome screening (QRFP)
Assay data:1 Tested
SummaryRelated BioAssays by Target
GPR103 Eurofins-Panlabs selectivity data (BI)
Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cell membrane by TopCount scintillation counter method
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization at 10 uM preincubated for 30 mins followed by agonist addition measured after 3 mins by Fluo-4 AM-based scanning fluorometery
Assay data:1 Active, 2 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization at 100 uM preincubated for 15 mins followed by agonist addition measured after 3 mins by Fluo-4 AM-based scanning fluorometery relative to 26RFa (20 to 26 residues)
Assay data:3 Tested
Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubated for 15 mins followed by agonist addition measured after 3 mins by Fluo-4 AM-based scanning fluorometery
Assay data:3 Active, 1 Activity ≤ 1 µM, 35 Tested
Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based scanning fluorometery
Assay data:9 Active, 3 Activity ≤ 1 µM, 36 Tested
Human QRFP receptor (QRFP receptor)
Assay data:6 Active, 6 Tested
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced TNF-alpha response in human macrophages_Primary screen TNF readout
Assay data:2853 Active, 18113 Tested
SummaryRelated BioAssays by Same Project
Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation counting
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assay
Assay data:12 Active, 9 Activity ≤ 1 µM, 14 Tested
A screen to identify synthetic lethal interactions with E-cadherin in an MCF10A isogenic cell line
Assay data:2442 Active, 18052 Tested
SummaryPubMed Citation
A screen to identify genes that regulate lymphatic endothelial cell migration - Primary Screen
Assay data:1034 Active, 18120 Tested
SummaryRelated BioAssays by Depositor
Identification of proteins required for the processing of the EWS-FLI1 nascent transcript
Assay data:59220 Tested
Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation counting
Assay data:19 Active, 10 Activity ≤ 1 µM, 22 Tested
Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assay
Assay data:25 Active, 15 Activity ≤ 1 µM, 30 Tested
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