BioAssay by Target (List) for Gene (Select 7443) - PubChem BioAssay - NCBI

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Select item 19126101.

Thermal Shift Assay. Domain: start/stop: R3-D336

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:27 Tested

AID:: 1912610

Summary Related BioAssays by Target

Select item 18353322.

VRK1 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1835332

Summary Related BioAssays by Target

Select item 18352013.

VRK1(h) Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1835201

Summary Related BioAssays by Target

Select item 18343704.

Inhibition of VRK1 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1834370

Summary PubMed Citation Related BioAssays by Target

Select item 17938495.

VRK1(VRK1LGRI) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793849

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17935656.

VRK1(VRK1LGRI) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793565

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17932717.

VRK1(VRK1LGRI) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793271

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17924998.

VRK1 ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1792499

Summary Related BioAssays by Target

Select item 17895039.

VRK1(h) Eurofins Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1789503

Summary Related BioAssays by Target

Select item 178755910.

VRK1(h) Millipore kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1787559

Summary Related BioAssays by Target

Select item 174960511.

Inhibition of VRK1 (unknown origin) assessed as residual activity measured at 1 uM

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:3 Tested

AID:: 1749605

Summary Related BioAssays by Target

Select item 171618712.

Inhibition of VRK1 (unknown origin) assessed as residual activity at 1 uM by Kinomescan method relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1716187

Summary PubMed Citation Related BioAssays by Target

Select item 171546713.

Inhibition of human VRK1 assessed as residual activity using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate at 1 uM by [gamma-33P]-ATP assay relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1715467

Summary PubMed Citation Related BioAssays by Target

Select item 167950114.

Inhibition of human VRK1 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate assessed as residual activity at 1 uM by [gamma-33P]-ATP assay relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:2 Tested

AID:: 1679501

Summary PubMed Citation Related BioAssays by Target

Select item 160884115.

Inhibition of recombinant human VRK1 at 1 uM incubated for 40 mins in presence of [gamma-33P]-ATP by scintillation counting method relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1608841

Summary PubMed Citation Related BioAssays by Target

Select item 160642416.

Inhibition of VRK1 (unknown origin) at 1 uM relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1606424

Summary PubMed Citation Related BioAssays by Target

Select item 158112717.

Inhibition of human VRK1 in presence of 10 uM ATP by radiometric analysis

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1581127

Summary PubMed Citation Related BioAssays by Target

Select item 158062518.

Inhibition of human VRK1 at 10 uM by radiometric assay relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1580625

Summary PubMed Citation Related BioAssays by Target

Select item 157959019.

Inhibition of human VRK1 at 1 uM by radiometric method relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1579590

Summary PubMed Citation Related BioAssays by Target

Select item 156869920.

Inhibition of human VRK1 at 100 nM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase VRK1

Assay data:1 Tested

AID:: 1568699

Summary PubMed Citation Related BioAssays by Target

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Target

RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (4)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 µM (6)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (10)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (43)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (44)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (1)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (33)
BioAssays extracted from the literature
NIH MLP (1)
BioAssays deposited by the NIH Molecular Libraries Program
Other (52)
BioAssays deposited by other experimentalists

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