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Binding affinity to mouse adenosine A2A receptor expressed in human HEK293 cell membrane by radioligand inhibition assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells at 10 uM incubated for 60 mins by radioligand binding assay
Assay data:3 Tested
Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
FLIPR and cAMP Inhibition Assay from US Patent US10858365: "Triazolo-pyrimidine compounds and uses thereof"
Assay data:117 Active, 13 Activity ≤ 1 nM, 116 Activity ≤ 1 µM, 119 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Displacement of [3H]CGS21680 from mouse A2A receptor expressed in HEK293 cells at 10 uM by radio ligand binding assay relative to control
Assay data:5 Tested
Antagonist activity at adenosine 2A receptor in BALB/c mouse T cells assessed as reduction in CGS-21680-induced suppression of IFN-gamma secretion incubated for 24 hrs by ELISA
Antagonist activity at adenosine 2A receptor in BALB/c mouse T cells assessed as reduction in CGS-21680-induced suppression of IL-2 secretion incubated for 24 hrs by ELISA
Antagonist activity at recombinant mouse A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assay
Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by scintillation proximity assay
Assay data:4 Active, 2 Activity ≤ 1 µM, 4 Tested
Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by scintillation proximity assay relative to adenosine 5-N-ethyluronamide
Assay data:7 Tested
Displacement of [3H]ZM241385 from mouse A2A receptor at 10 uM
Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method
Assay data:2 Tested
Displacement of [3H]ZM241385 from recombinant mouse adenosine receptor A2A expressed in HEK293 cell membranes after 1 hr by FACS analysis
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Mouse A2A receptor (Adenosine receptors)
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced NF-kappaB and TNF-alpha responses in mouse macrophages_Primary screen NFkB readout
Assay data:762 Active, 16821 Tested
SummaryRelated BioAssays by Same Project
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced NF-kappaB and TNF-alpha responses in mouse macrophages_Primary screen TNF readout
Assay data:1106 Active, 16821 Tested
Displacement of [3H]CGS21680 from mouse A2A adenosine receptor expressed in HEK293 cells at 10 uM after 60 mins by liquid scintillation counting
Antagonist activity at adenosine A2A receptor in C57/BL6 mouse lymphocytes assessed as inhibition of CGS-21680-mediated cAMP accumulation at 0.5 to 10 uM after 15 mins by ELISA
Assay data:2 Active, 2 Tested
Antagonist activity at adenosine A2A receptor in C57/BL6 mouse lymphocytes assessed as inhibition of CGS-21680-mediated cAMP accumulation after 15 mins by ELISA
Assay data:1 Active, 1 Tested
A screen to identify the genes that modify the response of osteosarcoma to doxorubicin in mouse - Primary Screen
Assay data:788 Active, 16789 Tested
SummaryPubMed Citation
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